
OpenAlex is a bibliographic catalogue of scientific papers, authors and institutions accessible in open access mode, named after the Library of Alexandria. It's citation coverage is excellent and I hope you will find utility in this listing of citing articles!
If you click the article title, you'll navigate to the article, as listed in CrossRef. If you click the Open Access links, you'll navigate to the "best Open Access location". Clicking the citation count will open this listing for that article. Lastly at the bottom of the page, you'll find basic pagination options.
Requested Article:
Biased Receptor Signaling in Drug Discovery
Terry Kenakin
Pharmacological Reviews (2019) Vol. 71, Iss. 2, pp. 267-315
Open Access | Times Cited: 246
Terry Kenakin
Pharmacological Reviews (2019) Vol. 71, Iss. 2, pp. 267-315
Open Access | Times Cited: 246
Showing 1-25 of 246 citing articles:
TRUPATH, an open-source biosensor platform for interrogating the GPCR transducerome
Reid H. J. Olsen, Jeffrey F. DiBerto, Justin G. English, et al.
Nature Chemical Biology (2020) Vol. 16, Iss. 8, pp. 841-849
Open Access | Times Cited: 423
Reid H. J. Olsen, Jeffrey F. DiBerto, Justin G. English, et al.
Nature Chemical Biology (2020) Vol. 16, Iss. 8, pp. 841-849
Open Access | Times Cited: 423
Review of the Endocannabinoid System
Hui‐Chen Lu, Ken Mackie
Biological Psychiatry Cognitive Neuroscience and Neuroimaging (2020) Vol. 6, Iss. 6, pp. 607-615
Open Access | Times Cited: 355
Hui‐Chen Lu, Ken Mackie
Biological Psychiatry Cognitive Neuroscience and Neuroimaging (2020) Vol. 6, Iss. 6, pp. 607-615
Open Access | Times Cited: 355
Virtual discovery of melatonin receptor ligands to modulate circadian rhythms
Reed M. Stein, Hye Jin Kang, John D. McCorvy, et al.
Nature (2020) Vol. 579, Iss. 7800, pp. 609-614
Open Access | Times Cited: 276
Reed M. Stein, Hye Jin Kang, John D. McCorvy, et al.
Nature (2020) Vol. 579, Iss. 7800, pp. 609-614
Open Access | Times Cited: 276
Molecular basis of β-arrestin coupling to formoterol-bound β1-adrenoceptor
Yang Lee, Tony Warne, Rony Nehmé, et al.
Nature (2020) Vol. 583, Iss. 7818, pp. 862-866
Open Access | Times Cited: 233
Yang Lee, Tony Warne, Rony Nehmé, et al.
Nature (2020) Vol. 583, Iss. 7818, pp. 862-866
Open Access | Times Cited: 233
GPCR activation mechanisms across classes and macro/microscales
Alexander S. Hauser, Albert J. Kooistra, Christian Munk, et al.
Nature Structural & Molecular Biology (2021) Vol. 28, Iss. 11, pp. 879-888
Open Access | Times Cited: 183
Alexander S. Hauser, Albert J. Kooistra, Christian Munk, et al.
Nature Structural & Molecular Biology (2021) Vol. 28, Iss. 11, pp. 879-888
Open Access | Times Cited: 183
Effector membrane translocation biosensors reveal G protein and βarrestin coupling profiles of 100 therapeutically relevant GPCRs
Charlotte Avet, Arturo Mancini, Billy Breton, et al.
eLife (2022) Vol. 11
Open Access | Times Cited: 177
Charlotte Avet, Arturo Mancini, Billy Breton, et al.
eLife (2022) Vol. 11
Open Access | Times Cited: 177
Psychedelics in Psychiatry: Neuroplastic, Immunomodulatory, and Neurotransmitter Mechanisms
Antonio Inserra, Danilo De Gregorio, Gabriella Gobbi
Pharmacological Reviews (2020) Vol. 73, Iss. 1, pp. 202-277
Open Access | Times Cited: 156
Antonio Inserra, Danilo De Gregorio, Gabriella Gobbi
Pharmacological Reviews (2020) Vol. 73, Iss. 1, pp. 202-277
Open Access | Times Cited: 156
Community guidelines for GPCR ligand bias: IUPHAR review 32
Peter Kolb, Terry Kenakin, S P H Alexander, et al.
British Journal of Pharmacology (2022) Vol. 179, Iss. 14, pp. 3651-3674
Open Access | Times Cited: 153
Peter Kolb, Terry Kenakin, S P H Alexander, et al.
British Journal of Pharmacology (2022) Vol. 179, Iss. 14, pp. 3651-3674
Open Access | Times Cited: 153
Common coupling map advances GPCR-G protein selectivity
Alexander S. Hauser, Charlotte Avet, Claire Normand, et al.
eLife (2022) Vol. 11
Open Access | Times Cited: 105
Alexander S. Hauser, Charlotte Avet, Claire Normand, et al.
eLife (2022) Vol. 11
Open Access | Times Cited: 105
GPCR kinase knockout cells reveal the impact of individual GRKs on arrestin binding and GPCR regulation
Julia Drube, Raphael S. Haider, Edda S. F. Matthees, et al.
Nature Communications (2022) Vol. 13, Iss. 1
Open Access | Times Cited: 83
Julia Drube, Raphael S. Haider, Edda S. F. Matthees, et al.
Nature Communications (2022) Vol. 13, Iss. 1
Open Access | Times Cited: 83
Identification of 5-HT2A receptor signaling pathways associated with psychedelic potential
Jason Wallach, Andrew B. Cao, Maggie M. Calkins, et al.
Nature Communications (2023) Vol. 14, Iss. 1
Open Access | Times Cited: 44
Jason Wallach, Andrew B. Cao, Maggie M. Calkins, et al.
Nature Communications (2023) Vol. 14, Iss. 1
Open Access | Times Cited: 44
Direct interrogation of context-dependent GPCR activity with a universal biosensor platform
Remi Janicot, Marcin Maziarz, Jong‐Chan Park, et al.
Cell (2024) Vol. 187, Iss. 6, pp. 1527-1546.e25
Open Access | Times Cited: 19
Remi Janicot, Marcin Maziarz, Jong‐Chan Park, et al.
Cell (2024) Vol. 187, Iss. 6, pp. 1527-1546.e25
Open Access | Times Cited: 19
Targeting cryptic allosteric sites of G protein-coupled receptors as a novel strategy for biased drug discovery
Xin Qiao, Xiaolong Li, Mingyang Zhang, et al.
Pharmacological Research (2025) Vol. 212, pp. 107574-107574
Open Access | Times Cited: 1
Xin Qiao, Xiaolong Li, Mingyang Zhang, et al.
Pharmacological Research (2025) Vol. 212, pp. 107574-107574
Open Access | Times Cited: 1
Combinatorial expression of GPCR isoforms affects signalling and drug responses
Maria Martí-Solano, Stephanie E. Crilly, Duccio Malinverni, et al.
Nature (2020) Vol. 587, Iss. 7835, pp. 650-656
Open Access | Times Cited: 112
Maria Martí-Solano, Stephanie E. Crilly, Duccio Malinverni, et al.
Nature (2020) Vol. 587, Iss. 7835, pp. 650-656
Open Access | Times Cited: 112
Pharmacology of Free Fatty Acid Receptors and Their Allosteric Modulators
Manuel Grundmann, Eckhard Bender, Jens Schamberger, et al.
International Journal of Molecular Sciences (2021) Vol. 22, Iss. 4, pp. 1763-1763
Open Access | Times Cited: 95
Manuel Grundmann, Eckhard Bender, Jens Schamberger, et al.
International Journal of Molecular Sciences (2021) Vol. 22, Iss. 4, pp. 1763-1763
Open Access | Times Cited: 95
A Biased View of μ-Opioid Receptors?
Alexandra E. Conibear, Eamonn Kelly
Molecular Pharmacology (2019) Vol. 96, Iss. 5, pp. 542-549
Open Access | Times Cited: 94
Alexandra E. Conibear, Eamonn Kelly
Molecular Pharmacology (2019) Vol. 96, Iss. 5, pp. 542-549
Open Access | Times Cited: 94
Neurobiology of cannabinoid receptor signaling
Beat Lutz
Dialogues in Clinical Neuroscience (2020) Vol. 22, Iss. 3, pp. 207-222
Open Access | Times Cited: 79
Beat Lutz
Dialogues in Clinical Neuroscience (2020) Vol. 22, Iss. 3, pp. 207-222
Open Access | Times Cited: 79
G protein-coupled receptor-G protein interactions: a single-molecule perspective
Davide Calebiro, Zsombor Kőszegi, Yann Lanoiselée, et al.
Physiological Reviews (2020) Vol. 101, Iss. 3, pp. 857-906
Open Access | Times Cited: 78
Davide Calebiro, Zsombor Kőszegi, Yann Lanoiselée, et al.
Physiological Reviews (2020) Vol. 101, Iss. 3, pp. 857-906
Open Access | Times Cited: 78
The Interplay of Glucagon-Like Peptide-1 Receptor Trafficking and Signalling in Pancreatic Beta Cells
Amaara Marzook, Alejandra Tomás, Ben Jones
Frontiers in Endocrinology (2021) Vol. 12
Open Access | Times Cited: 67
Amaara Marzook, Alejandra Tomás, Ben Jones
Frontiers in Endocrinology (2021) Vol. 12
Open Access | Times Cited: 67
The G protein database, GproteinDb
Gáspár Pándy‐Szekeres, Mauricio Esguerra, Alexander S. Hauser, et al.
Nucleic Acids Research (2021) Vol. 50, Iss. D1, pp. D518-D525
Open Access | Times Cited: 65
Gáspár Pándy‐Szekeres, Mauricio Esguerra, Alexander S. Hauser, et al.
Nucleic Acids Research (2021) Vol. 50, Iss. D1, pp. D518-D525
Open Access | Times Cited: 65
Biased Agonism: Lessons from Studies of Opioid Receptor Agonists
Eamonn Kelly, Alexandra E. Conibear, Graeme Henderson
The Annual Review of Pharmacology and Toxicology (2022) Vol. 63, Iss. 1, pp. 491-515
Open Access | Times Cited: 44
Eamonn Kelly, Alexandra E. Conibear, Graeme Henderson
The Annual Review of Pharmacology and Toxicology (2022) Vol. 63, Iss. 1, pp. 491-515
Open Access | Times Cited: 44
Selective activation of Gαob by an adenosine A1 receptor agonist elicits analgesia without cardiorespiratory depression
Mark J. Wall, Emily Hill, Robert Huckstepp, et al.
Nature Communications (2022) Vol. 13, Iss. 1
Open Access | Times Cited: 43
Mark J. Wall, Emily Hill, Robert Huckstepp, et al.
Nature Communications (2022) Vol. 13, Iss. 1
Open Access | Times Cited: 43
In-cell NMR: Why and how?
François‐Xavier Theillet, Enrico Luchinat
Progress in Nuclear Magnetic Resonance Spectroscopy (2022) Vol. 132-133, pp. 1-112
Open Access | Times Cited: 38
François‐Xavier Theillet, Enrico Luchinat
Progress in Nuclear Magnetic Resonance Spectroscopy (2022) Vol. 132-133, pp. 1-112
Open Access | Times Cited: 38
The application of artificial intelligence to accelerate G protein‐coupled receptor drug discovery
Thi Nguyen, Diep Thi Ngoc Nguyen, Huan Yee Koh, et al.
British Journal of Pharmacology (2023) Vol. 181, Iss. 14, pp. 2371-2384
Open Access | Times Cited: 22
Thi Nguyen, Diep Thi Ngoc Nguyen, Huan Yee Koh, et al.
British Journal of Pharmacology (2023) Vol. 181, Iss. 14, pp. 2371-2384
Open Access | Times Cited: 22
Specific pharmacological and Gi/o protein responses of some native GPCRs in neurons
Chanjuan Xu, Yiwei Zhou, Yuxuan Liu, et al.
Nature Communications (2024) Vol. 15, Iss. 1
Open Access | Times Cited: 8
Chanjuan Xu, Yiwei Zhou, Yuxuan Liu, et al.
Nature Communications (2024) Vol. 15, Iss. 1
Open Access | Times Cited: 8