Open Access Helper

OpenAlex Citation Counts

OpenAlex Citations Logo

OpenAlex is a bibliographic catalogue of scientific papers, authors and institutions accessible in open access mode, named after the Library of Alexandria. It's citation coverage is excellent and I hope you will find utility in this listing of citing articles!

If you click the article title, you'll navigate to the article, as listed in CrossRef. If you click the Open Access links, you'll navigate to the "best Open Access location". Clicking the citation count will open this listing for that article. Lastly at the bottom of the page, you'll find basic pagination options.

Requested Article:

Signalling bias in new drug discovery: detection, quantification and therapeutic impact
Terry Kenakin, Arthur Christopoulos
Nature Reviews Drug Discovery (2012) Vol. 12, Iss. 3, pp. 205-216
Open Access | Times Cited: 684

Showing 1-25 of 684 citing articles:

Molecular Dynamics Simulation for All
Scott A. Hollingsworth, Ron O. Dror
Neuron (2018) Vol. 99, Iss. 6, pp. 1129-1143
Open Access | Times Cited: 1935
Structure-based discovery of opioid analgesics with reduced side effects
Aashish Manglik, Henry J. Lin, Dipendra K. Aryal, et al.
Nature (2016) Vol. 537, Iss. 7619, pp. 185-190
Open Access | Times Cited: 869
Biased signalling: from simple switches to allosteric microprocessors
Jeffrey S. Smith, Robert J. Lefkowitz, Sudarshan Rajagopal
Nature Reviews Drug Discovery (2018) Vol. 17, Iss. 4, pp. 243-260
Open Access | Times Cited: 643
Allosteric sodium in class A GPCR signaling
Vsevolod Katritch, Gustavo Fenalti, Enrique E. Abola, et al.
Trends in Biochemical Sciences (2014) Vol. 39, Iss. 5, pp. 233-244
Open Access | Times Cited: 465
Muscarinic acetylcholine receptors: novel opportunities for drug development
Andrew C. Kruse, Brian K. Kobilka, Dinesh Gautam, et al.
Nature Reviews Drug Discovery (2014) Vol. 13, Iss. 7, pp. 549-560
Open Access | Times Cited: 389
The Diverse Roles of Arrestin Scaffolds in G Protein–Coupled Receptor Signaling
Yuri K. Peterson, Louis M. Luttrell
Pharmacological Reviews (2017) Vol. 69, Iss. 3, pp. 256-297
Open Access | Times Cited: 377
Structure of the Nanobody-Stabilized Active State of the Kappa Opioid Receptor
Tao Che, Susruta Majumdar, Saheem A. Zaidi, et al.
Cell (2018) Vol. 172, Iss. 1-2, pp. 55-67.e15
Open Access | Times Cited: 338
Biased ligands at G-protein-coupled receptors: promise and progress
Jonathan D. Violin, Aimee L. Crombie, David G. Soergel, et al.
Trends in Pharmacological Sciences (2014) Vol. 35, Iss. 7, pp. 308-316
Closed Access | Times Cited: 336
The experimental power of FR900359 to study Gq-regulated biological processes
Ramona Schrage, Anna-Lena Schmitz, Evelyn Gaffal, et al.
Nature Communications (2015) Vol. 6, Iss. 1
Open Access | Times Cited: 322
Glucagon-Like Peptide-1 and Its Class B G Protein–Coupled Receptors: A Long March to Therapeutic Successes
Chris de Graaf, Dan Donnelly, Denise Wootten, et al.
Pharmacological Reviews (2016) Vol. 68, Iss. 4, pp. 954-1013
Open Access | Times Cited: 315
Structure and function of serotonin G protein-coupled receptors
John D. McCorvy, Bryan L. Roth
Pharmacology & Therapeutics (2015) Vol. 150, pp. 129-142
Open Access | Times Cited: 312
The role of kinetic context in apparent biased agonism at GPCRs
Carmen Klein Herenbrink, David A. Sykes, Prashant Donthamsetti, et al.
Nature Communications (2016) Vol. 7, Iss. 1
Open Access | Times Cited: 312
Cannabinoid CB2 receptor ligand profiling reveals biased signalling and off-target activity
Marjolein Soethoudt, Uwe Grether, Jürgen Fingerle, et al.
Nature Communications (2017) Vol. 8, Iss. 1
Open Access | Times Cited: 305
Allosteric Modulation as a Unifying Mechanism for Receptor Function and Regulation
Jean‐Pierre Changeux, Arthur Christopoulos
Cell (2016) Vol. 166, Iss. 5, pp. 1084-1102
Open Access | Times Cited: 285
Recent developments in biased agonism
James W. Wisler, Kunhong Xiao, A. Thomsen, et al.
Current Opinion in Cell Biology (2013) Vol. 27, pp. 18-24
Open Access | Times Cited: 272
Structure of the Adenosine A1 Receptor Reveals the Basis for Subtype Selectivity
Alisa Glukhova, David M. Thal, Thi Nguyen, et al.
Cell (2017) Vol. 168, Iss. 5, pp. 867-877.e13
Open Access | Times Cited: 270
Biased agonism: An emerging paradigm in GPCR drug discovery
Zoran Ranković, Tarsis F. Brust, Laura Bohn
Bioorganic & Medicinal Chemistry Letters (2015) Vol. 26, Iss. 2, pp. 241-250
Open Access | Times Cited: 248
Distinct profiles of functional discrimination among G proteins determine the actions of G protein–coupled receptors
Ikuo Masuho, Olga Ostrovskaya, Grant M. Kramer, et al.
Science Signaling (2015) Vol. 8, Iss. 405
Open Access | Times Cited: 245
Nanobodies to Study G Protein–Coupled Receptor Structure and Function
Aashish Manglik, Brian K. Kobilka, Jan Steyaert
The Annual Review of Pharmacology and Toxicology (2016) Vol. 57, Iss. 1, pp. 19-37
Open Access | Times Cited: 244
The Pharmacology and Function of Receptors for Short-Chain Fatty Acids
Daniele Bolognini, Andrew B. Tobin, Graeme Milligan, et al.
Molecular Pharmacology (2015) Vol. 89, Iss. 3, pp. 388-398
Open Access | Times Cited: 242
Opportunities and challenges in the discovery of allosteric modulators of GPCRs for treating CNS disorders
P. Jeffrey Conn, Craig W. Lindsley, Jens Meiler, et al.
Nature Reviews Drug Discovery (2014) Vol. 13, Iss. 9, pp. 692-708
Open Access | Times Cited: 239
International Union of Basic and Clinical Pharmacology. XC. Multisite Pharmacology: Recommendations for the Nomenclature of Receptor Allosterism and Allosteric Ligands
Arthur Christopoulos, Jean‐Pierre Changeux, William A. Catterall, et al.
Pharmacological Reviews (2014) Vol. 66, Iss. 4, pp. 918-947
Open Access | Times Cited: 223
Quantification of Ligand Bias for Clinically Relevant β2-Adrenergic Receptor Ligands: Implications for Drug Taxonomy
Emma T. van der Westhuizen, Billy Breton, Arthur Christopoulos, et al.
Molecular Pharmacology (2013) Vol. 85, Iss. 3, pp. 492-509
Closed Access | Times Cited: 223
Allosteric Modulation of GPCRs: New Insights and Potential Utility for Treatment of Schizophrenia and Other CNS Disorders
Daniel J. Foster, P. Jeffrey Conn
Neuron (2017) Vol. 94, Iss. 3, pp. 431-446
Open Access | Times Cited: 218
Advances in G Protein-Coupled Receptor Allostery: From Function to Structure
Arthur Christopoulos
Molecular Pharmacology (2014) Vol. 86, Iss. 5, pp. 463-478
Open Access | Times Cited: 213
Page 1 - Next Page

Scroll to top