
OpenAlex is a bibliographic catalogue of scientific papers, authors and institutions accessible in open access mode, named after the Library of Alexandria. It's citation coverage is excellent and I hope you will find utility in this listing of citing articles!
If you click the article title, you'll navigate to the article, as listed in CrossRef. If you click the Open Access links, you'll navigate to the "best Open Access location". Clicking the citation count will open this listing for that article. Lastly at the bottom of the page, you'll find basic pagination options.
Requested Article:
Chamelogk: A Chromatographic Chameleonicity Quantifier to Design Orally Bioavailable Beyond-Rule-of-5 Drugs
Diego García Jiménez, Maura Vallaro, Matteo Rossi Sebastiano, et al.
Journal of Medicinal Chemistry (2023) Vol. 66, Iss. 15, pp. 10681-10693
Open Access | Times Cited: 18
Diego García Jiménez, Maura Vallaro, Matteo Rossi Sebastiano, et al.
Journal of Medicinal Chemistry (2023) Vol. 66, Iss. 15, pp. 10681-10693
Open Access | Times Cited: 18
Showing 18 citing articles:
Beyond Rule of Five and PROTACs in Modern Drug Discovery: Polarity Reducers, Chameleonicity, and the Evolving Physicochemical Landscape
Edward Price, Manuel Weinheimer, Alexey Rivkin, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 7, pp. 5683-5698
Closed Access | Times Cited: 23
Edward Price, Manuel Weinheimer, Alexey Rivkin, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 7, pp. 5683-5698
Closed Access | Times Cited: 23
Exploring the chemical space of orally bioavailable PROTACs
Giulia Apprato, Vasanthanathan Poongavanam, Diego García Jiménez, et al.
Drug Discovery Today (2024) Vol. 29, Iss. 4, pp. 103917-103917
Open Access | Times Cited: 15
Giulia Apprato, Vasanthanathan Poongavanam, Diego García Jiménez, et al.
Drug Discovery Today (2024) Vol. 29, Iss. 4, pp. 103917-103917
Open Access | Times Cited: 15
Molecular chameleons in drug discovery
Vasanthanathan Poongavanam, Lianne H. E. Wieske, Stefan Peintner, et al.
Nature Reviews Chemistry (2023) Vol. 8, Iss. 1, pp. 45-60
Closed Access | Times Cited: 27
Vasanthanathan Poongavanam, Lianne H. E. Wieske, Stefan Peintner, et al.
Nature Reviews Chemistry (2023) Vol. 8, Iss. 1, pp. 45-60
Closed Access | Times Cited: 27
Use of Aldehyde–Alkyne–Amine Couplings to Generate Medicinal Chemistry-Relevant Linkers
Andrew McGown, Vesna Vetma, Damien Crépin, et al.
ACS Medicinal Chemistry Letters (2025)
Open Access
Andrew McGown, Vesna Vetma, Damien Crépin, et al.
ACS Medicinal Chemistry Letters (2025)
Open Access
Targeted protein degradation in CNS disorders: a promising route to novel therapeutics?
Sandra Kuemper, Andrew G. Cairns, Kristian Birchall, et al.
Frontiers in Molecular Neuroscience (2024) Vol. 17
Open Access | Times Cited: 6
Sandra Kuemper, Andrew G. Cairns, Kristian Birchall, et al.
Frontiers in Molecular Neuroscience (2024) Vol. 17
Open Access | Times Cited: 6
IMHB-Mediated Chameleonicity in Drug Design: A Focus on Structurally Related PROTACs
Diego García Jiménez, Matteo Rossi Sebastiano, Maura Vallaro, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 13, pp. 11421-11434
Closed Access | Times Cited: 5
Diego García Jiménez, Matteo Rossi Sebastiano, Maura Vallaro, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 13, pp. 11421-11434
Closed Access | Times Cited: 5
Assessment of the Efficiency of Selecting Promising Compounds During Virtual Screening Based on Various Estimations of Drug-Likeness
Vladislav S. Sukhachev, Alexander V. Dmitriev, Sergey M. Ivanov, et al.
Pharmaceutical Chemistry Journal (2025)
Closed Access
Vladislav S. Sukhachev, Alexander V. Dmitriev, Sergey M. Ivanov, et al.
Pharmaceutical Chemistry Journal (2025)
Closed Access
Finding a needle in the haystack: ADME and pharmacokinetics/pharmacodynamics characterization and optimization toward orally available bifunctional protein degraders
Giulia Apprato, Giulia Caron, Gauri Deshmukh, et al.
Expert Opinion on Drug Discovery (2025)
Closed Access
Giulia Apprato, Giulia Caron, Gauri Deshmukh, et al.
Expert Opinion on Drug Discovery (2025)
Closed Access
Computational approaches to aid PROTAC drug discovery
Sohini Chakraborti, Kirsten McAulay
Elsevier eBooks (2025)
Closed Access
Sohini Chakraborti, Kirsten McAulay
Elsevier eBooks (2025)
Closed Access
Molecular properties, including chameleonicity, as essential tools for designing the next generation of oral beyond rule of five drugs
Giulia Caron, Diego García Jiménez, Maura Vallaro, et al.
ADMET & DMPK (2024)
Open Access | Times Cited: 3
Giulia Caron, Diego García Jiménez, Maura Vallaro, et al.
ADMET & DMPK (2024)
Open Access | Times Cited: 3
Conquering the beyond Rule of Five Space with an Optimized High-Throughput Caco-2 Assay to Close Gaps in Absorption Prediction
Patricia Muschong, Khader Awwad, Edward Price, et al.
Pharmaceutics (2024) Vol. 16, Iss. 7, pp. 846-846
Open Access | Times Cited: 2
Patricia Muschong, Khader Awwad, Edward Price, et al.
Pharmaceutics (2024) Vol. 16, Iss. 7, pp. 846-846
Open Access | Times Cited: 2
To homeostasis and beyond! Recent advances in the medicinal chemistry of heterobifunctional derivatives
Diana Castagna, Benoit Gourdet, Roland Hjerpe, et al.
Progress in medicinal chemistry (2024), pp. 61-160
Closed Access | Times Cited: 1
Diana Castagna, Benoit Gourdet, Roland Hjerpe, et al.
Progress in medicinal chemistry (2024), pp. 61-160
Closed Access | Times Cited: 1
Chromatographic Determination of Permeability-Relevant Lipophilicity Facilitates Rapid Analysis of Macrocyclic Peptide Scaffolds
Grant Koch, Åke Engström, Jaru Taechalertpaisarn, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 21, pp. 19612-19622
Open Access | Times Cited: 1
Grant Koch, Åke Engström, Jaru Taechalertpaisarn, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 21, pp. 19612-19622
Open Access | Times Cited: 1
Meeting report: DMPK optimisation strategies and quantitative translational PKPD frameworks to predict human PK and efficacious dose of targeted protein degraders
Caroline Rynn, Heide Marika Duevel
Xenobiotica (2024) Vol. 54, Iss. 9, pp. 776-780
Closed Access
Caroline Rynn, Heide Marika Duevel
Xenobiotica (2024) Vol. 54, Iss. 9, pp. 776-780
Closed Access
Molecular Transformers: Adaptive Multitarget Ligands for Esterase-Induced Transition from Analgesics to Anesthetics
Tianguang Huang, Chi Song, Yuhao Chen, et al.
Journal of Medicinal Chemistry (2024)
Closed Access
Tianguang Huang, Chi Song, Yuhao Chen, et al.
Journal of Medicinal Chemistry (2024)
Closed Access
A novel application of Hydrophilic Interaction Liquid Chromatography for the identification of compounds with intramolecular hydrogen bonds.
Alessandra Pugliano, Bernd Kuhn, Nenad Manevski, et al.
Journal of Pharmaceutical and Biomedical Analysis (2024) Vol. 252, pp. 116499-116499
Closed Access
Alessandra Pugliano, Bernd Kuhn, Nenad Manevski, et al.
Journal of Pharmaceutical and Biomedical Analysis (2024) Vol. 252, pp. 116499-116499
Closed Access
Closing the Design–Make–Test–Analyze Loop: Interplay between Experiments and Predictions Drives PROTACs Bioavailability
Zulma Santisteban Valencia, Jennifer Kingston, Filip Miljković, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 22, pp. 20242-20257
Closed Access
Zulma Santisteban Valencia, Jennifer Kingston, Filip Miljković, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 22, pp. 20242-20257
Closed Access
Exploring the Potential of Adaptive, Local Machine Learning in Comparison to the Prediction Performance of Global Models: A Case Study from Bayer’s Caco-2 Permeability Database
Frank Filip Steinbauer, Thorsten Lehr, Andreas Reichel
Journal of Chemical Information and Modeling (2024)
Open Access
Frank Filip Steinbauer, Thorsten Lehr, Andreas Reichel
Journal of Chemical Information and Modeling (2024)
Open Access