
OpenAlex is a bibliographic catalogue of scientific papers, authors and institutions accessible in open access mode, named after the Library of Alexandria. It's citation coverage is excellent and I hope you will find utility in this listing of citing articles!
If you click the article title, you'll navigate to the article, as listed in CrossRef. If you click the Open Access links, you'll navigate to the "best Open Access location". Clicking the citation count will open this listing for that article. Lastly at the bottom of the page, you'll find basic pagination options.
Requested Article:
A Versatile and Sustainable Multicomponent Platform for the Synthesis of Protein Degraders: Proof-of-Concept Application to BRD4-Degrading PROTACs
Irene Preet Bhela, Alice Ranza, Federica Carolina Balestrero, et al.
Journal of Medicinal Chemistry (2022) Vol. 65, Iss. 22, pp. 15282-15299
Open Access | Times Cited: 33
Irene Preet Bhela, Alice Ranza, Federica Carolina Balestrero, et al.
Journal of Medicinal Chemistry (2022) Vol. 65, Iss. 22, pp. 15282-15299
Open Access | Times Cited: 33
Showing 1-25 of 33 citing articles:
Accelerating Drug Discovery: Synthesis of Complex Chemotypes via Multicomponent Reactions
Melissa J. Buskes, Aaron Coffin, Dawn M. Troast, et al.
ACS Medicinal Chemistry Letters (2023) Vol. 14, Iss. 4, pp. 376-385
Open Access | Times Cited: 44
Melissa J. Buskes, Aaron Coffin, Dawn M. Troast, et al.
ACS Medicinal Chemistry Letters (2023) Vol. 14, Iss. 4, pp. 376-385
Open Access | Times Cited: 44
Advancing Strategies for Proteolysis-Targeting Chimera Design
Minglei Li, Ying Zhi, Bo Liu, et al.
Journal of Medicinal Chemistry (2023) Vol. 66, Iss. 4, pp. 2308-2329
Closed Access | Times Cited: 43
Minglei Li, Ying Zhi, Bo Liu, et al.
Journal of Medicinal Chemistry (2023) Vol. 66, Iss. 4, pp. 2308-2329
Closed Access | Times Cited: 43
Current advances and development strategies of orally bioavailable PROTACs
Shenxin Zeng, Yingqiao Ye, Heye Xia, et al.
European Journal of Medicinal Chemistry (2023) Vol. 261, pp. 115793-115793
Closed Access | Times Cited: 33
Shenxin Zeng, Yingqiao Ye, Heye Xia, et al.
European Journal of Medicinal Chemistry (2023) Vol. 261, pp. 115793-115793
Closed Access | Times Cited: 33
A beginner’s guide to current synthetic linker strategies towards VHL-recruiting PROTACs
Nikol A. Zografou-Barredo, Alex J. Hallatt, J. S. JUN. RICCI, et al.
Bioorganic & Medicinal Chemistry (2023) Vol. 88-89, pp. 117334-117334
Open Access | Times Cited: 30
Nikol A. Zografou-Barredo, Alex J. Hallatt, J. S. JUN. RICCI, et al.
Bioorganic & Medicinal Chemistry (2023) Vol. 88-89, pp. 117334-117334
Open Access | Times Cited: 30
PROTACs: A novel strategy for cancer drug discovery and development
Xin Han, Yi Sun
MedComm (2023) Vol. 4, Iss. 3
Open Access | Times Cited: 24
Xin Han, Yi Sun
MedComm (2023) Vol. 4, Iss. 3
Open Access | Times Cited: 24
Innovative, combinatorial and high-throughput approaches to degrader synthesis
Rebecca Stevens, James D. F. Thompson, Julie C. L. Fournier, et al.
Chemical Society Reviews (2024) Vol. 53, Iss. 10, pp. 4838-4861
Closed Access | Times Cited: 9
Rebecca Stevens, James D. F. Thompson, Julie C. L. Fournier, et al.
Chemical Society Reviews (2024) Vol. 53, Iss. 10, pp. 4838-4861
Closed Access | Times Cited: 9
Accelerating PROTACs Discovery Through a Direct‐to‐Biology Platform Enabled by Modular Photoclick Chemistry
Ke‐Nian Yan, Yong‐Qiang Nie, Jiayu Wang, et al.
Advanced Science (2024) Vol. 11, Iss. 26
Open Access | Times Cited: 7
Ke‐Nian Yan, Yong‐Qiang Nie, Jiayu Wang, et al.
Advanced Science (2024) Vol. 11, Iss. 26
Open Access | Times Cited: 7
Rapid PROTAC Discovery Platform: Nanomole-Scale Array Synthesis and Direct Screening of Reaction Mixtures
Mateusz P. Plesniak, Emilia K. Taylor, Frederik Eisele, et al.
ACS Medicinal Chemistry Letters (2023) Vol. 14, Iss. 12, pp. 1882-1890
Closed Access | Times Cited: 18
Mateusz P. Plesniak, Emilia K. Taylor, Frederik Eisele, et al.
ACS Medicinal Chemistry Letters (2023) Vol. 14, Iss. 12, pp. 1882-1890
Closed Access | Times Cited: 18
Targeted protein degradation: advances in drug discovery and clinical practice
Guangcai Zhong, Xiaoyu Chang, Weilin Xie, et al.
Signal Transduction and Targeted Therapy (2024) Vol. 9, Iss. 1
Open Access | Times Cited: 6
Guangcai Zhong, Xiaoyu Chang, Weilin Xie, et al.
Signal Transduction and Targeted Therapy (2024) Vol. 9, Iss. 1
Open Access | Times Cited: 6
Novel SK channel positive modulators prevent ferroptosis and excitotoxicity in neuronal cells
Yuequ Zhang, Shabnam Shaabani, Kirsty Vowinkel, et al.
Biomedicine & Pharmacotherapy (2024) Vol. 171, pp. 116163-116163
Open Access | Times Cited: 5
Yuequ Zhang, Shabnam Shaabani, Kirsty Vowinkel, et al.
Biomedicine & Pharmacotherapy (2024) Vol. 171, pp. 116163-116163
Open Access | Times Cited: 5
Perspectives on Nuclear Magnetic Resonance Spectroscopy in Drug Discovery Research
Janet Caceres‐Cortes, Bradley T. Falk, Luciano Mueller, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 3, pp. 1701-1733
Closed Access | Times Cited: 5
Janet Caceres‐Cortes, Bradley T. Falk, Luciano Mueller, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 3, pp. 1701-1733
Closed Access | Times Cited: 5
Use of Aldehyde–Alkyne–Amine Couplings to Generate Medicinal Chemistry-Relevant Linkers
Andrew McGown, Vesna Vetma, Damien Crépin, et al.
ACS Medicinal Chemistry Letters (2025)
Open Access
Andrew McGown, Vesna Vetma, Damien Crépin, et al.
ACS Medicinal Chemistry Letters (2025)
Open Access
Versatile One-Pot Synthesis of Hydrophobic Tags by Multicomponent Reactions
Federica Carolina Balestrero, Laura Gioiello, Georgia Goutsiou, et al.
ACS Omega (2025) Vol. 10, Iss. 5, pp. 4745-4753
Open Access
Federica Carolina Balestrero, Laura Gioiello, Georgia Goutsiou, et al.
ACS Omega (2025) Vol. 10, Iss. 5, pp. 4745-4753
Open Access
Instant Macrocyclizations via Multicomponent Reactions
Michael Fragkiadakis, Paraskevi-Kleio Anastasiou, Marios Zingiridis, et al.
The Journal of Organic Chemistry (2023) Vol. 88, Iss. 17, pp. 12709-12715
Closed Access | Times Cited: 8
Michael Fragkiadakis, Paraskevi-Kleio Anastasiou, Marios Zingiridis, et al.
The Journal of Organic Chemistry (2023) Vol. 88, Iss. 17, pp. 12709-12715
Closed Access | Times Cited: 8
A one-pot photocatalytic triazole-based linkerology for PROTACs
Jinhua Liu, Yaqi Deng, Jiabin Yin, et al.
Cell Reports Physical Science (2024) Vol. 5, Iss. 8, pp. 102139-102139
Open Access | Times Cited: 2
Jinhua Liu, Yaqi Deng, Jiabin Yin, et al.
Cell Reports Physical Science (2024) Vol. 5, Iss. 8, pp. 102139-102139
Open Access | Times Cited: 2
PROTAC unleashed: Unveiling the synthetic approaches and potential therapeutic applications
Narayanaperumal Pravin, Krzysztof Jóźwiak
European Journal of Medicinal Chemistry (2024) Vol. 279, pp. 116837-116837
Open Access | Times Cited: 2
Narayanaperumal Pravin, Krzysztof Jóźwiak
European Journal of Medicinal Chemistry (2024) Vol. 279, pp. 116837-116837
Open Access | Times Cited: 2
Next steps for targeted protein degradation
Mackenzie W. Krone, Craig M. Crews
Cell chemical biology (2024)
Closed Access | Times Cited: 2
Mackenzie W. Krone, Craig M. Crews
Cell chemical biology (2024)
Closed Access | Times Cited: 2
A practical “preTACs-cytoblot” platform accelerates the streamlined development of PROTAC-based protein degraders
Zijian Rao, Kailin Li, Ju-Eun Hong, et al.
European Journal of Medicinal Chemistry (2023) Vol. 251, pp. 115248-115248
Closed Access | Times Cited: 7
Zijian Rao, Kailin Li, Ju-Eun Hong, et al.
European Journal of Medicinal Chemistry (2023) Vol. 251, pp. 115248-115248
Closed Access | Times Cited: 7
Regioselective Access to 1,2,4-Triazole-Fused N-Heterocycle, Pyrrolo[1,2-a][1,2,4]triazolo[5,1-c]pyrazine, via Double Dehydrative Cyclizations
Hyunjin Oh, Hye‐Yeon Kim, Ikyon Kim
The Journal of Organic Chemistry (2023) Vol. 88, Iss. 16, pp. 11748-11761
Closed Access | Times Cited: 7
Hyunjin Oh, Hye‐Yeon Kim, Ikyon Kim
The Journal of Organic Chemistry (2023) Vol. 88, Iss. 16, pp. 11748-11761
Closed Access | Times Cited: 7
One-Pot Synthesis of Cereblon Proteolysis Targeting Chimeras via Photoinduced C(sp2)–C(sp3) Cross Coupling and Amide Formation for Proteolysis Targeting Chimera Library Synthesis
Christine Marie Arndt, Jacqueline Bitai, Jessica Brunner, et al.
Journal of Medicinal Chemistry (2023) Vol. 66, Iss. 24, pp. 16939-16952
Closed Access | Times Cited: 7
Christine Marie Arndt, Jacqueline Bitai, Jessica Brunner, et al.
Journal of Medicinal Chemistry (2023) Vol. 66, Iss. 24, pp. 16939-16952
Closed Access | Times Cited: 7
Accessing three-branched high-affinity cereblon ligands for molecular glue and protein degrader design
Robert D. Kuchta, Christopher Heim, Alexander Herrmann, et al.
RSC Chemical Biology (2023) Vol. 4, Iss. 3, pp. 229-234
Open Access | Times Cited: 6
Robert D. Kuchta, Christopher Heim, Alexander Herrmann, et al.
RSC Chemical Biology (2023) Vol. 4, Iss. 3, pp. 229-234
Open Access | Times Cited: 6
Late-stage synthesis of heterobifunctional molecules for PROTAC applications via ruthenium-catalysed C‒H amidation
Daniele Antermite, Stig D. Friis, Johan R. Johansson, et al.
Nature Communications (2023) Vol. 14, Iss. 1
Open Access | Times Cited: 6
Daniele Antermite, Stig D. Friis, Johan R. Johansson, et al.
Nature Communications (2023) Vol. 14, Iss. 1
Open Access | Times Cited: 6
A Tunable Cascade Reaction of Ureidomalonates and Alkenyl Azlactones for the Divergent Synthesis of Hydantoins with Distinct Functional Groups
Lin Chen, Di Wang
The Journal of Organic Chemistry (2024) Vol. 89, Iss. 5, pp. 3365-3382
Closed Access | Times Cited: 1
Lin Chen, Di Wang
The Journal of Organic Chemistry (2024) Vol. 89, Iss. 5, pp. 3365-3382
Closed Access | Times Cited: 1
Hijacking the MDM2 E3 Ligase with novel BRD4-Targeting PROTACs in Pancreatic Cancer Cells
Mihaela P. Ficu, Dan Niculescu‐Duvaz, Mohammed Aljarah, et al.
(2024)
Open Access | Times Cited: 1
Mihaela P. Ficu, Dan Niculescu‐Duvaz, Mohammed Aljarah, et al.
(2024)
Open Access | Times Cited: 1
To homeostasis and beyond! Recent advances in the medicinal chemistry of heterobifunctional derivatives
Diana Castagna, Benoit Gourdet, Roland Hjerpe, et al.
Progress in medicinal chemistry (2024), pp. 61-160
Closed Access | Times Cited: 1
Diana Castagna, Benoit Gourdet, Roland Hjerpe, et al.
Progress in medicinal chemistry (2024), pp. 61-160
Closed Access | Times Cited: 1