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OpenAlex is a bibliographic catalogue of scientific papers, authors and institutions accessible in open access mode, named after the Library of Alexandria. It's citation coverage is excellent and I hope you will find utility in this listing of citing articles!

If you click the article title, you'll navigate to the article, as listed in CrossRef. If you click the Open Access links, you'll navigate to the "best Open Access location". Clicking the citation count will open this listing for that article. Lastly at the bottom of the page, you'll find basic pagination options.

Requested Article:

Novel pyrazolo-tetrahydropyridines as potent orexin receptor antagonists
Thierry Sifferlen, Christoph Boss, Emmanuelle Cottreel, et al.
Bioorganic & Medicinal Chemistry Letters (2010) Vol. 20, Iss. 5, pp. 1539-1542
Closed Access | Times Cited: 17

Showing 17 citing articles:

Discovery of the Dual Orexin Receptor Antagonist [(7R)-4-(5-Chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl]methanone (MK-4305) for the Treatment of Insomnia
Christopher D. Cox, Michael J. Breslin, David B. Whitman, et al.
Journal of Medicinal Chemistry (2010) Vol. 53, Iss. 14, pp. 5320-5332
Closed Access | Times Cited: 348
Selective orexin receptor antagonists
Terry P. Lebold, Pascal Bonaventure, Brock T. Shireman
Bioorganic & Medicinal Chemistry Letters (2013) Vol. 23, Iss. 17, pp. 4761-4769
Closed Access | Times Cited: 73
The Use of Physiology-Based Pharmacokinetic and Pharmacodynamic Modeling in the Discovery of the Dual Orexin Receptor Antagonist ACT-541468
Alexander Treiber, Ruben de Kanter, Catherine Roch, et al.
Journal of Pharmacology and Experimental Therapeutics (2017) Vol. 362, Iss. 3, pp. 489-503
Open Access | Times Cited: 69
Substituted pyrrolidin-2-ones: Centrally acting orexin receptor antagonists promoting sleep. Part 2
Thierry Sifferlen, Amandine Boller, Audrey Chardonneau, et al.
Bioorganic & Medicinal Chemistry Letters (2015) Vol. 25, Iss. 9, pp. 1884-1891
Closed Access | Times Cited: 31
Acyl Meldrum's acid derivatives: application in organic synthesis
Karolina Janikowska, Janusz Rachoń, Sławomir Makowiec
Russian Chemical Reviews (2014) Vol. 83, Iss. 7, pp. 620-637
Closed Access | Times Cited: 20
Discovery of Highly Potent Dual Orexin Receptor Antagonists via a Scaffold‐Hopping Approach
Bibia Heidmann, John Gatfield, Catherine Roch, et al.
ChemMedChem (2016) Vol. 11, Iss. 19, pp. 2132-2146
Closed Access | Times Cited: 17
Discovery of substituted lactams as novel dual orexin receptor antagonists. Synthesis, preliminary structure–activity relationship studies and efforts towards improved metabolic stability and pharmacokinetic properties. Part 1
Thierry Sifferlen, Amandine Boller, Audrey Chardonneau, et al.
Bioorganic & Medicinal Chemistry Letters (2014) Vol. 24, Iss. 4, pp. 1201-1208
Closed Access | Times Cited: 16
Bio-based triacetic acid lactone in the synthesis of azaheterocyclesviaa ring-opening transformation
Дмитрий Л. Обыденнов, Asmaa I. El-Tantawy, Vyacheslav Ya. Sosnovskikh
New Journal of Chemistry (2018) Vol. 42, Iss. 11, pp. 8943-8952
Closed Access | Times Cited: 15
Structure–activity relationship studies and sleep-promoting activity of novel 1-chloro-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine derivatives as dual orexin receptor antagonists. Part 2
Thierry Sifferlen, Ralf Koberstein, Emmanuelle Cottreel, et al.
Bioorganic & Medicinal Chemistry Letters (2013) Vol. 23, Iss. 13, pp. 3857-3863
Closed Access | Times Cited: 13
Synthesis, structure–activity relationship studies, and identification of novel 5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine derivatives as dual orexin receptor antagonists. Part 1
Thierry Sifferlen, Ralf Koberstein, Emmanuelle Cottreel, et al.
Bioorganic & Medicinal Chemistry Letters (2013) Vol. 23, Iss. 7, pp. 2212-2216
Closed Access | Times Cited: 11
Oxadiazole Derivatives as Dual Orexin Receptor Antagonists: Synthesis, Structure–Activity Relationships, and Sleep‐Promoting Properties in Rats
Christine Brotschi, Catherine Roch, John Gatfield, et al.
ChemMedChem (2019) Vol. 14, Iss. 13, pp. 1257-1270
Closed Access | Times Cited: 10
Discovery and optimisation of 1-acyl-2-benzylpyrrolidines as potent dual orexin receptor antagonists
Jodi T. Williams, John Gatfield, Catherine Roch, et al.
MedChemComm (2015) Vol. 6, Iss. 6, pp. 1054-1064
Closed Access | Times Cited: 9
Discovery of novel tetrahydro-pyrazolo [4,3-c] pyridines for the treatment of neuropathic pain: Synthesis and neuropharmacology
Perumal Yogeeswari, Monika Sharma, Ganesh Samala, et al.
European Journal of Medicinal Chemistry (2013) Vol. 66, pp. 211-220
Closed Access | Times Cited: 9
From Oxadiazole to Triazole Analogues: Optimization toward a Dual Orexin Receptor Antagonist with Improved in vivo Efficacy in Dogs
Christine Brotschi, Martin H. Bolli, John Gatfield, et al.
ChemMedChem (2020) Vol. 15, Iss. 5, pp. 430-448
Closed Access | Times Cited: 6
The halogensulfonylative cyclizations of 1,6-enynes with sodium sulfinate/TBAX for the regioselective synthesis of tetrahydropyridines
Tian-Meng Kang, Yiwen Wu, Wenshu Zheng, et al.
Tetrahedron (2023) Vol. 135, pp. 133339-133339
Closed Access | Times Cited: 1
Orexin Receptor Antagonists
Brock T. Shireman, Michael A. Letavic
Elsevier eBooks (2016), pp. 225-279
Closed Access | Times Cited: 1
ChemInform Abstract: Novel Pyrazolo‐tetrahydropyridines as Potent Orexin Receptor Antagonists
Thierry Sifferlen, Christoph Boss, Emmanuelle Cottreel, et al.
ChemInform (2010) Vol. 41, Iss. 29
Closed Access
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